SCHEMBL8304633

SCHEMBL8304633

COc1ccc(N)cc1C1CCN(CCCCCCCCCCCCCCCC(F)(F)F)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
HTR4 Q13639 7/20 0.43
ACHE P22303 2/20 0.43
CHRM2 P08172 2/20 0.40
CHRM4 P08173 2/20 0.40
CHRM5 P08912 2/20 0.40
CHRM1 P11229 2/20 0.40
CHRM3 P20309 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CACNA1G O43497 1/20 0.38
KCNH2 Q12809 1/20 0.38
ADORA2A P29274 1/20 0.38
ABCB1 P08183 1/20 0.38
GRM2 Q14416 2/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6784774 0.85 DRD2 (0.55) DRD2HTR4ACHECHRM4CHRM5
SCHEMBL7029357 0.76 QDPR (0.52) DRD2MEN1KMT2AKDM4E
SCHEMBL7938441 0.73 KDM4E (0.46) KDM4EADRA1A
SCHEMBL6646479 0.73 DRD2 (0.52) DRD2MEN1KMT2AADRA1DADRA1A
SCHEMBL6815771 0.72 MEN1 (0.45) MEN1KMT2AKCNH2
SCHEMBL8304631 0.72 HTR4 (0.36) DRD2HTR4ACHEMEN1KMT2A
SCHEMBL7880812 0.72 HTR2A (0.47)
SCHEMBL6924205 0.72 ABCB1 (0.43) DRD2CHRM2CHRM4CHRM5CHRM1
SCHEMBL14320526 0.72 SIGMAR1 (0.46) DRD2MEN1KMT2A
SCHEMBL6717514 0.71 EHMT2 (0.42) DRD2MEN1KMT2AKDM4EKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0898569-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GmbH (DE) 1999-03-03 EP disclosed
WO-1997040038-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GMBH (DE) 1997-10-30 WO disclosed