SCHEMBL8305196

SCHEMBL8305196

CCC(Nc1ccncc1)C1CCCN(C2CCC(CC(=O)O)CC2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
KDM4E B2RXH2 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ADRA1A P35348 3/20 0.34
HSD11B1 P28845 1/20 0.34
KCNH2 Q12809 3/20 0.33
IDH1 O75874 2/20 0.33
CHRM1 P11229 1/20 0.33
DAPK3 O43293 1/20 0.33
ROCK2 O75116 1/20 0.33
CHEK2 O96017 1/20 0.33
PIM1 P11309 1/20 0.33
PLK1 P53350 1/20 0.33
ROCK1 Q13464 1/20 0.33
CDC42BPA Q5VT25 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301327 0.73 KDM4E (0.43) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8300331 0.71 KDM4E (0.43) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8304375 0.69 ITGB3 (0.43) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8298652 0.68 ITGB3 (0.45) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8300030 0.68 KDM4E (0.45) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8615087 0.67 ITGB3 (0.36) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8613755 0.67 ITGB3 (0.56) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8300686 0.66 NAMPT (0.43) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8300507 0.66 KDM4E (0.43) ITGB3ITGA2BKDM4EKMT2AMEN1
SCHEMBL8304879 0.65 KDM4E (0.42) ITGB3ITGA2BKDM4EKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed
EP-0808306-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1997-11-26 EP disclosed
WO-1996024586-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1996-08-15 WO disclosed