SCHEMBL8305404

SCHEMBL8305404

CCCCCCCCOc1cc2c(c(F)n1)CC(c1ncc(O)cn1)CC2

nearest known ligand 0.32

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.32
DRD1 P21728 10/20 0.31
DRD3 P35462 8/20 0.31
CNR1 P21554 2/20 0.31
CNR2 P34972 2/20 0.31
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
TAOK3 Q9H2K8 1/20 0.31
PTPN1 P18031 1/20 0.30
DRD2 P14416 1/20 0.30
HTR3E A5X5Y0 1/20 0.30
HTR3B O95264 1/20 0.30
HTR3A P46098 1/20 0.30
HTR3D Q70Z44 1/20 0.30
HTR3C Q8WXA8 1/20 0.30
NR5A1 Q13285 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305524 0.91 HTR1D (0.33) GPR84HTR1AHTR1DHTR1BTAOK3
SCHEMBL8303039 0.87 NR5A1 (0.33) DRD1DRD3CNR1CNR2TAOK3
SCHEMBL8298273 0.78 GPR84 (0.34) GPR84CNR1CNR2TAOK3HTR3E
SCHEMBL8293978 0.78 CNR2 (0.32) GPR84CNR1CNR2
SCHEMBL8301428 0.70 THRA (0.34) GPR84CNR1CNR2TAOK3HTR3E
SCHEMBL8299252 0.70 NR5A1 (0.32) GPR84CNR1CNR2HTR3EHTR3B
SCHEMBL5722827 0.69 HTR1D (0.33) DRD1DRD3CNR1CNR2HTR1D
SCHEMBL8296395 0.69 THRA (0.32) GPR84CNR1CNR2TAOK3
SCHEMBL8294020 0.69 THRA (0.38) GPR84CNR1CNR2TAOK3HTR3E
SCHEMBL8305593 0.65 XDH (0.40) HTR1DHTR1BNR5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824520-B1 1-FLUOR-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES AND THEIR USE IN LIQUID CRYSTAL MIXTURES HOECHST AG (DE) 1999-10-06 EP disclosed
US-5942618-A 3,7-DISUBSTITUTED 1-FLUORO-5,6,7,8-TETRAHYDROISOQUINOLINE DERIVATIVES HAVING EXCELLENT LIGHT, CHEMICAL AND THERMAL STABILITY; COLORLESS IN PURE STATE; USE IN SWITCHING AND/OR DISPLAY DEVICE HOECHST AKTIENGESELLSCHAFT (DE) 1999-08-24 US disclosed