SCHEMBL8307133

SCHEMBL8307133

COCCN(C)S(=O)(=O)c1ccc2c(c1)C(Cl)(Cl)C(=O)N2

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 3/20 0.63
PKLR P30613 1/20 0.45
GAA P10253 2/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
VCAM1 P19320 3/20 0.39
ALDH1A1 P00352 2/20 0.37
GSTO1 P78417 1/20 0.37
MAOA P21397 2/20 0.37
MAOB P27338 1/20 0.37
MAPT P10636 1/20 0.36
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950459 0.85 KMT2A (0.48) CASP3PKLRGAAVCAM1ALDH1A1
SCHEMBL6946269 0.82 PKLR (0.44) CASP3PKLRGAAVCAM1ALDH1A1
SCHEMBL6949029 0.79 PKLR (0.42) CASP3PKLRGAAALDH1A1MAOA
SCHEMBL6535335 0.78 CASP3 (1.00) CASP3GAAALDH1A1MAOAMAOB
SCHEMBL6943633 0.78 ALDH1A1 (0.58) PKLRGAAALDH1A1MAPTLMNA
SCHEMBL8307129 0.77 PKLR (0.50) PKLRGAAVCAM1ALDH1A1MAPT
SCHEMBL8307006 0.75 PKLR (0.42) CASP3PKLRGAAALDH1A1MAOA
SCHEMBL3917930 0.71 SIGMAR1 (0.55) CASP3ALDH1A1GSTO1MAPTLMNA
SCHEMBL1368050 0.71 CASP3 (0.54) CASP3GAAPTGDR2VCAM1ALDH1A1
SCHEMBL30555219 0.71 PKLR (0.55) PKLRGAAALDH1A1MAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed