SCHEMBL8308786

SCHEMBL8308786

Cc1c(C2CCN(c3ccc(Cl)cc3)CC2)n[nH]c1-c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 8/20 0.43
DRD2 P14416 6/20 0.43
DRD3 P35462 6/20 0.43
CETP P11597 1/20 0.42
MAPK13 O15264 2/20 0.40
MAPK12 P53778 2/20 0.40
MAPK11 Q15759 2/20 0.40
MAPK14 Q16539 2/20 0.40
SLC9A1 P19634 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
TSHR P16473 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LMNA P02545 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
AVPR1A P37288 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388392 0.84 DRD4 (0.60) DRD4DRD2DRD3ALDH1A1CYP1A2
SCHEMBL1388702 0.81 DRD4 (0.66) DRD4DRD2DRD3ALDH1A1CYP1A2
SCHEMBL6974758 0.76 DRD2 (0.36) DRD4DRD2DRD3MAPK13MAPK12
SCHEMBL6974762 0.76 LCAT (0.37) DRD4DRD2DRD3MAPK13MAPK12
SCHEMBL1388459 0.71 ALDH1A1 (0.45) DRD4DRD2DRD3ALDH1A1LMNA
SCHEMBL1388772 0.70 TRPV6 (0.47) DRD4DRD2DRD3ALDH1A1TSHR
SCHEMBL31612521 0.70 MEN1 (0.61) DRD4DRD2ALDH1A1CYP1A2LMNA
SCHEMBL15657195 0.69 GRM5 (0.40) DRD4DRD2DRD3ALDH1A1CYP1A2
SCHEMBL1388752 0.68 SIGMAR1 (0.55) DRD4DRD2DRD3ALDH1A1CYP1A2
SCHEMBL23630311 0.68 ALDH1A1 (0.43) DRD4DRD2DRD3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665833-B1 DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME (GB) 1999-07-14 EP claimed