SCHEMBL8313790

SCHEMBL8313790

CC1(C)C=C(c2ccccn2)c2cc(C#N)ccc2OC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
METAP2 P50579 1/20 0.39
METAP1 P53582 1/20 0.39
GRM5 P41594 15/20 0.37
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313018 0.91 METAP2 (0.39) TGFBR1MAPK13MAPK12MAPK11MAPK14
SCHEMBL8332841 0.83 METAP2 (0.40) TGFBR1MAPK13MAPK12MAPK11MAPK14
SCHEMBL8315486 0.83 NPC1 (0.39) TGFBR1METAP2METAP1GRM5KDM4E
SCHEMBL8312863 0.82 MAPT (0.39) TGFBR1METAP2METAP1GRM5KDM4E
SCHEMBL8315585 0.82 ADRA1A (0.40) METAP1GRM5KDM4EMAPTHTT
SCHEMBL8314584 0.82 FABP6 (0.37) TGFBR1MAPK14METAP2METAP1GRM5
SCHEMBL8311893 0.82 MAOA (0.35) TGFBR1MAPK13MAPK12MAPK11MAPK14
SCHEMBL8315902 0.82 MAOA (0.33) TGFBR1MAPK13MAPK12MAPK11MAPK14
SCHEMBL8316184 0.81 KDM4E (0.37) METAP1KDM4EALDH1A1MAPTHTT
SCHEMBL8310381 0.81 HTR2B (0.40) TGFBR1GRM5KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed