SCHEMBL8315347

SCHEMBL8315347

COc1ccc(C=CC(=O)NC2CCCNC(=O)C2)cc1OCCSC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.46
MAPT P10636 2/20 0.45
PDE4B Q07343 2/20 0.45
ALDH1A1 P00352 4/20 0.43
RAB9A P51151 2/20 0.43
LMNA P02545 1/20 0.43
MMP2 P08253 1/20 0.42
KDM4E B2RXH2 1/20 0.41
FDPS P14324 1/20 0.41
CNR2 P34972 1/20 0.41
HDAC3 O15379 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
HDAC4 P56524 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
HDAC1 Q13547 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313606 0.88 TP53 (0.56) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8311933 0.83 ALDH1A1 (0.49) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8313214 0.82 TP53 (0.47) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8312845 0.82 RECQL (0.54) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8317573 0.80 KMT2A (0.52) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8317248 0.78 PTGS2 (0.52) TP53MAPTALDH1A1RAB9AHDAC3
SCHEMBL8312914 0.76 TP53 (0.53) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8312438 0.76 PTGS2 (0.45) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8314971 0.76 MAOB (0.48) TP53MAPTALDH1A1RAB9ALMNA
SCHEMBL8311715 0.76 L3MBTL1 (0.53) MAPTPDE4BALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0351856-B1 Thiazolo[5,4-b]azepine compounds TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-09-15 EP disclosed
US-4956360-A LIPOPEROXIDE INHIBITORS, ENZYME INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-09-11 US disclosed