SCHEMBL8315724

SCHEMBL8315724

CC(C)N1Cc2cccc(C(F)(F)F)c2N(CCCl)S1(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.35
ACACB O00763 2/20 0.35
MC4R P32245 1/20 0.33
AADAT Q8N5Z0 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
DRD3 P35462 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318169 0.84 SLC6A2 (0.34) MC4RALDH1A1DRD3KCNH2
SCHEMBL8317987 0.83 ADRA2A (0.36) ACACBMC4RAADATKDM4EALDH1A1
SCHEMBL8315238 0.82 P2RX7 (0.33) P2RX7AADATKDM4E
SCHEMBL8318057 0.77 KDM4E (0.39) KDM4E
SCHEMBL8316061 0.72 CRY1 (0.35) KCNH2
SCHEMBL8314015 0.72 SLC6A2 (0.39) KDM4EDRD3KCNH2
SCHEMBL8316696 0.68 SLC6A2 (0.38) KDM4E
SCHEMBL6985168 0.68 HTR2A (0.40) KDM4E
SCHEMBL6982495 0.67 KCNH2 (0.32) KCNH2
SCHEMBL7081764 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929072-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY LIMITED (GB) 1999-07-27 US disclosed
EP-0897921-A1 Benzothiadiazinyl-indole derivatives and their use as serotonin receptor ligands ELI LILLY AND COMPANY LIMITED (GB) 1999-02-24 EP disclosed