SCHEMBL8319432

SCHEMBL8319432

O=C(O)[C@H]1C[C@H]2CCC[C@H]2N1S(=O)(=O)c1ccc(-c2ccc([N+](=O)[O-])cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.52
MMP2 P08253 2/20 0.45
FAAH O00519 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
EPHX2 P34913 1/20 0.43
AKR1C3 P42330 1/20 0.40
MMP8 P22894 8/20 0.40
MMP3 P08254 5/20 0.40
MMP1 P03956 1/20 0.40
MMP7 P09237 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2961151 1.00 ACHE (0.52) ACHEMMP2FAAHCA1CA2
SCHEMBL13201349 0.98 ACHE (0.49) ACHEMMP2FAAHCA1CA2
SCHEMBL8328565 0.96 ACHE (0.55) ACHEMMP2FAAHEPHX2AKR1C3
SCHEMBL2965640 0.96 ACHE (0.55) ACHEMMP2FAAHEPHX2AKR1C3
SCHEMBL13201328 0.88 CA9 (0.52) ACHEMMP2CA1CA2CA9
SCHEMBL8319435 0.87 MMP2 (0.48) ACHEMMP2CA1CA2CA9
SCHEMBL2959199 0.85 AKR1C3 (0.39) MMP2AKR1C3MMP8MMP3MMP1
SCHEMBL16298352 0.85 AKR1C3 (0.39) MMP2AKR1C3MMP8MMP3MMP1
SCHEMBL8319047 0.85 PSEN1 (0.52) ACHEAKR1C3MMP8MMP3
SCHEMBL8319431 0.85 AKR1C3 (0.39) MMP2AKR1C3MMP8MMP3MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7772270-B2 Imino acid derivatives as inhibitors of matrix metalloproteinases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2010-08-10 US disclosed
US-7772270-B2 Imino acid derivatives as inhibitors of matrix metalloproteinases SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2010-08-10 US disclosed
WO-2004060874-A1 IMINO ACID DERIVATIVES FOR USE AS INHIBITORS OF MATRIX METALLOPROTEINASES AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-07-22 WO disclosed