SCHEMBL8323194

SCHEMBL8323194

Nc1cccc([CH]CC(N)c2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.50
MAOB P27338 3/20 0.50
CYP19A1 P11511 2/20 0.50
NPSR1 Q6W5P4 1/20 0.40
SCN4A P35499 4/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
GFER P55789 1/20 0.38
CPN1 P15169 1/20 0.37
CPB2 Q96IY4 1/20 0.37
TACR1 P25103 2/20 0.36
CYP3A4 P08684 1/20 0.35
CASP1 P29466 1/20 0.35
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322584 0.82 MAOA (0.49) MAOAMAOBCYP19A1NPSR1NPC1
SCHEMBL8324378 0.82 SCN4A (0.44) SCN4ANPC1TACR1
SCHEMBL8321946 0.82 NFE2L2 (0.49) NPC1CYP3A4
SCHEMBL8324064 0.82 SCN4A (0.44) MAOBSCN4ANPC1TACR1
SCHEMBL8326302 0.82 HTR2A (0.41) SCN4A
SCHEMBL8322926 0.78 IDO1 (0.52) NPC1MAPTTACR1
SCHEMBL8326846 0.77 RELA (0.46) SCN4ACYP3A4
SCHEMBL8327108 0.72 NFE2L2 (0.44) SCN4AMAPTRECQL
SCHEMBL8322049 0.72 TACR1 (0.41) SCN4ATACR1
SCHEMBL8326407 0.72 CYP3A4 (0.39) SCN4ANPC1TACR1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed