SCHEMBL8322926

SCHEMBL8322926

NC(C[CH]c1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.52
TDO2 P48775 2/20 0.52
TACR1 P25103 3/20 0.46
CACNA1F O60840 1/20 0.46
CACNA1D Q01668 1/20 0.46
CACNA1S Q13698 1/20 0.46
CACNA1C Q13936 1/20 0.46
PNMT P11086 1/20 0.44
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
ACP3 P15309 2/20 0.41
NFE2L2 Q16236 1/20 0.41
OPRM1 P35372 2/20 0.40
OPRD1 P41143 2/20 0.40
OPRK1 P41145 2/20 0.40
OPRL1 P41146 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322780 0.83 TACR1 (0.46) IDO1TDO2TACR1CACNA1FCACNA1D
SCHEMBL8324977 0.82 IDO1 (0.49) IDO1TDO2PNMTHTR2AHTR2C
SCHEMBL8321946 0.80 NFE2L2 (0.49) IDO1TDO2NFE2L2NPC1RAB9A
SCHEMBL8323194 0.78 MAOA (0.50) TACR1NPC1MAPT
SCHEMBL8324064 0.77 SCN4A (0.44) IDO1TDO2TACR1NPC1RAB9A
SCHEMBL8326302 0.77 HTR2A (0.41) HTR2A
SCHEMBL8324378 0.77 SCN4A (0.44) TACR1NPC1
SCHEMBL27796912 0.74 NFE2L2 (0.50) IDO1TDO2PNMTHTR2AHTR2C
SCHEMBL13358903 0.74 PNMT (0.51) IDO1TDO2TACR1PNMTHTR2A
SCHEMBL266165 0.74 PNMT (0.51) IDO1TDO2TACR1CACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed