SCHEMBL8323293

SCHEMBL8323293

COc1ccc(Oc2c(Cl)ncnc2Cl)cc1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
NPBWR1 P48145 2/20 0.46
MCHR1 Q99705 1/20 0.46
KDR P35968 1/20 0.43
LCK P06239 2/20 0.42
EGFR P00533 1/20 0.42
ALDH1A1 P00352 4/20 0.41
LMNA P02545 2/20 0.41
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41
TUBA1B P68363 2/20 0.41
TUBA4A P68366 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1748605 0.80 ALDH1A1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL8326548 0.80 CA12 (0.50) CA12CA1CA2CA7CA9
SCHEMBL7293817 0.79 ACHE (0.53) NPBWR1MCHR1EGFRALDH1A1SMN1; SMN2
SCHEMBL4435549 0.79 EDNRB (0.44) CA12CA1CA2CA7CA9
SCHEMBL7294631 0.78 ALDH1A1 (0.46) NPBWR1MCHR1LCKEGFRALDH1A1
SCHEMBL7298131 0.78 TRPA1 (0.45) PDGFRBPDGFRANPBWR1MCHR1KDR
SCHEMBL7303200 0.78 NPBWR1 (0.48) PDGFRBPDGFRANPBWR1MCHR1KDR
SCHEMBL1748457 0.77 DHPS (0.50) CA12CA1CA2CA7CA9
SCHEMBL8323843 0.77 CYP1A1 (0.47) NPBWR1MCHR1LCKALDH1A1LMNA
SCHEMBL8325304 0.76 ALDH1A1 (0.42) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0633259-B1 Sulfonylaminopyrimidines, their preparation and their use as medicine HOFFMANN LA ROCHE (CH) 1999-01-13 EP disclosed
US-5541186-A ENDOTHELIN RECEPTOR INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1996-07-30 US disclosed
EP-0633259-A1 Sulfonylaminopyrimidines, their preparation and their use as medicine F. HOFFMANN-LA ROCHE AG (CH) 1995-01-11 EP disclosed