SCHEMBL8324031

SCHEMBL8324031

COC(=O)/C=C/c1ccc(Cn2ccnc2-c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.47
ESR1 P03372 1/20 0.46
LIMK2 P53671 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 2/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
TYR P14679 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
KDM4E B2RXH2 1/20 0.43
IP6K1 Q92551 1/20 0.43
IP6K3 Q96PC2 1/20 0.43
IP6K2 Q9UHH9 1/20 0.43
HDAC1 Q13547 2/20 0.41
HDAC8 Q9BY41 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319277 0.86 HDAC1 (0.55) BRD4ESR1LIMK2HDAC1HDAC8
SCHEMBL8323972 0.79 BRD4 (0.43) BRD4SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL9485553 0.76 MMP1 (0.60) LIMK2SMN1; SMN2NPC1RAB9AKMT2A
SCHEMBL27706042 0.76 ESR1 (0.57) BRD4ESR1LIMK2SMN1; SMN2NPC1
SCHEMBL11050806 0.76 CA1 (0.51) BRD4ESR1LIMK2SMN1; SMN2NPC1
SCHEMBL8322937 0.76 CYP3A4 (0.49) SMN1; SMN2NPC1RAB9AKMT2ACA12
SCHEMBL17621 0.75 HSD17B10 (0.62) BRD4ESR1LIMK2KMT2ACYP1A2
SCHEMBL3439436 0.73 MEN1 (0.59) NPC1RAB9AKMT2AHDAC1HDAC8
SCHEMBL4833224 0.73 CA12 (0.66) ESR1SMN1; SMN2KMT2ACA12CA1
SCHEMBL4833218 0.73 CA12 (0.66) ESR1SMN1; SMN2KMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed