SCHEMBL8326191

SCHEMBL8326191

Fc1ccc([CH]CCc2ccccc2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
GPR52 Q9Y2T5 2/20 0.38
G6PC1 P35575 2/20 0.38
PLA2G1B P04054 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
EGFR P00533 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
MAPT P10636 1/20 0.35
NLRP3 Q96P20 1/20 0.35
CYP2A6 P11509 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3566359 0.84 G6PC1 (0.51) G6PC1SMN1; SMN2NPC1RAB9ANFKB1
SCHEMBL8324164 0.77 ALDH1A1 (0.51) SMN1; SMN2NPC1RAB9AMAPTTAAR1
SCHEMBL7814468 0.77 NFE2L2 (0.48) GPR52SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL28117454 0.74 TRPA1 (0.51) TRPA1PLA2G1BCYP1A2CYP3A4CYP2D6
SCHEMBL8325508 0.74 NFE2L2 (0.55) GPR52CYP1A2CYP3A4CYP2D6NPC1
SCHEMBL1115608 0.73 MAOB (0.46) GPR52SMN1; SMN2CYP2A6HTR2ATAAR1
SCHEMBL27692484 0.73 TRPA1 (0.46) TRPA1PLA2G1BCYP1A2CYP3A4CYP2D6
SCHEMBL27605856 0.73 TRPA1 (0.46) TRPA1PLA2G1BCYP1A2CYP3A4CYP2D6
SCHEMBL8326407 0.72 CYP3A4 (0.39) TRPA1PLA2G1BCYP1A2CYP3A4CYP2D6
SCHEMBL8327003 0.72 TRPA1 (0.38) TRPA1G6PC1CYP3A4CYP2D6NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed