SCHEMBL8327003

SCHEMBL8327003

CC([CH]c1ccc(F)c(Cl)c1)Cc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
PPARG P37231 2/20 0.37
PPARA Q07869 2/20 0.37
SLC6A2 P23975 3/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP3A4 P08684 1/20 0.36
KCNH2 Q12809 1/20 0.36
NOS2 P35228 1/20 0.36
LMNA P02545 1/20 0.36
TAAR1 Q96RJ0 5/20 0.36
SIGMAR1 Q99720 2/20 0.36
MAOA P21397 1/20 0.36
CYP2A6 P11509 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
PNMT P11086 1/20 0.35
G6PC1 P35575 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8322029 0.82 CYP3A4 (0.40) TRPA1PPARGPPARASLC6A2SLC6A4
SCHEMBL8323270 0.82 KDM4E (0.36) TRPA1PPARGPPARASLC6A2SLC6A4
SCHEMBL8319052 0.80 PNMT (0.49) SLC6A2SLC6A4SLC6A3LMNATAAR1
SCHEMBL8326594 0.78 NFE2L2 (0.44) TRPA1PPARGPPARASLC6A2SLC6A4
SCHEMBL8330718 0.77 NFE2L2 (0.49) PPARGPPARASLC6A2SLC6A4SLC6A3
SCHEMBL8327482 0.73 CYP3A4 (0.42) TRPA1SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL8327667 0.73 TAAR1 (0.44) TRPA1PPARGPPARASLC6A2SLC6A4
SCHEMBL8324318 0.72 TAAR1 (0.44) PPARGPPARASLC6A2SLC6A4SLC6A3
SCHEMBL8326191 0.72 TRPA1 (0.38) TRPA1CYP2D6CYP3A4TAAR1CYP2A6
SCHEMBL8323488 0.71 SLC6A2 (0.41) TRPA1PPARGPPARASLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed