SCHEMBL8326389

SCHEMBL8326389

COc1ccc(-c2ncc3c(n2)-c2cncnc2CC3)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
CCNB1 P14635 1/20 0.39
CCND1 P24385 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
CDK7 P50613 1/20 0.39
CDK9 P50750 1/20 0.39
CCNH P51946 1/20 0.39
PIK3CA P42336 2/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
CYP2A6 P11509 2/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
RPS6KA3 P51812 1/20 0.35
MAPKAPK2 P49137 3/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327878 0.84 CCNA2 (0.34) CDK2MAPKAPK2KDM4EALDH1A1
SCHEMBL8327052 0.82 CDK2 (0.35) CCNT1CDK1CDK4CCNB1CCND1
SCHEMBL8329431 0.79 CCNA2 (0.44) CDK2KDM4ECYP19A1
SCHEMBL8326151 0.78 CYP1A2 (0.41) CDK2CYP2A6KDM4EALDH1A1MAPT
SCHEMBL8327742 0.71 CCNA2 (0.34) CDK2KDM4EALDH1A1EGFR
SCHEMBL8325671 0.71 CCNA2 (0.40) CDK2KDM4E
SCHEMBL8325078 0.68 DUSP10 (0.47) CDK2MAPKAPK2KDM4EALDH1A1EGFR
SCHEMBL8327901 0.68 CCNA2 (0.46) CDK2MAPKAPK2KDM4EALDH1A1MAPT
SCHEMBL8328470 0.67 SLC22A12 (0.38) MAPKAPK2KDM4EALDH1A1CYP19A1SLC22A12
SCHEMBL8327012 0.65 CYP2A6 (0.46) CDK2CYP2A6KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP claimed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO claimed
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP disclosed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO disclosed