SCHEMBL8326463

SCHEMBL8326463

CCOC(=O)CC1(C(=O)OCC)Cn2c(cc3ccccc32)C1=O

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KDM4E B2RXH2 4/20 0.37
RAB9A P51151 1/20 0.37
OPRM1 P35372 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KMT2A Q03164 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GLA P06280 2/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
NOD2 Q9HC29 3/20 0.35
NOD1 Q9Y239 3/20 0.35
MEN1 O00255 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327585 0.89 OPRM1 (0.40) ALDH1A1KDM4ERAB9AOPRM1NPSR1
SCHEMBL8329097 0.77 OPRM1 (0.37) ALDH1A1KDM4EOPRM1KMT2AL3MBTL1
SCHEMBL8322854 0.75 ALDH1A1 (0.36) ALDH1A1KDM4ERAB9AOPRM1KMT2A
SCHEMBL8320925 0.75 HTR2A (0.42) ALDH1A1KDM4EOPRM1KMT2AGAA
SCHEMBL8330362 0.74 HTR2A (0.38) ALDH1A1KDM4ERAB9AOPRM1KMT2A
SCHEMBL8327931 0.74 NR1H2 (0.35) ALDH1A1OPRM1KMT2AL3MBTL1MEN1
SCHEMBL8328986 0.70 HTR2A (0.42) ALDH1A1KDM4ERAB9AOPRM1KMT2A
SCHEMBL8655802 0.68 MAPT (0.44) ALDH1A1KDM4ERAB9AKMT2AGAA
SCHEMBL7737588 0.68 ALDH1A1 (0.44) ALDH1A1KDM4EOPRM1NPSR1KMT2A
SCHEMBL30954226 0.67 ALDH1A1 (0.39) ALDH1A1KDM4ENPSR1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed