SCHEMBL8329097

SCHEMBL8329097

CCOC(=O)C1(CCC(=O)OC)CCn2c(cc3ccccc32)C1=O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
ALDH1A1 P00352 5/20 0.35
OPRD1 P41143 3/20 0.35
OPRK1 P41145 3/20 0.35
SLC22A1 O15245 1/20 0.35
SLC6A4 P31645 1/20 0.35
ADRA1A P35348 1/20 0.35
KCNH2 Q12809 1/20 0.35
CACNA1C Q13936 1/20 0.35
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327585 0.86 OPRM1 (0.40) OPRM1MEN1KMT2AALDH1A1OPRD1
SCHEMBL8327931 0.84 NR1H2 (0.35) OPRM1MEN1KMT2AALDH1A1OPRD1
SCHEMBL8326463 0.77 ALDH1A1 (0.40) OPRM1MEN1KMT2AALDH1A1KDM4E
SCHEMBL8327590 0.69 OPRM1 (0.35) OPRM1MEN1KMT2AALDH1A1OPRD1
SCHEMBL3156042 0.68 HTR2A (0.46) OPRM1OPRD1OPRK1SLC22A1SLC6A4
SCHEMBL8328986 0.66 HTR2A (0.42) OPRM1MEN1KMT2AALDH1A1OPRD1
SCHEMBL9344111 0.66 ALDH1A1 (0.42) OPRM1ALDH1A1OPRD1OPRK1SLC22A1
SCHEMBL8655802 0.64 MAPT (0.44) MEN1KMT2AALDH1A1KDM4E
SCHEMBL8325800 0.64 ALDH1A1 (0.39) MEN1KMT2AALDH1A1L3MBTL1LMNA
SCHEMBL8320925 0.64 HTR2A (0.42) OPRM1MEN1KMT2AALDH1A1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed