SCHEMBL8328181

SCHEMBL8328181

N#Cc1ccc(N(c2cncnc2)c2cc(F)ccc2F)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.38
GRM5 P41594 1/20 0.36
CYP3A4 P08684 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.34
VNN1 O95497 1/20 0.34
DPP4 P27487 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
DPP7 Q9UHL4 1/20 0.34
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33
ACLY P53396 1/20 0.33
NPY5R Q15761 1/20 0.33
KDM4E B2RXH2 1/20 0.32
TP53 P04637 1/20 0.32
PGR P06401 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330253 0.79 CYP19A1 (0.52) CYP19A1GRM5CYP3A4CYP11B1CYP11B2
SCHEMBL8326800 0.73 CYP19A1 (0.44) CYP19A1GRM5VNN1
SCHEMBL8324537 0.71 KIF11 (0.53) CYP19A1CYP3A4VNN1
SCHEMBL8324262 0.69 CYP19A1 (0.40) CYP19A1GRM5CYP3A4VNN1
SCHEMBL8323103 0.69 ESR1 (0.49) CYP19A1VNN1CYP11B1CYP11B2
SCHEMBL8327043 0.68 CYP19A1 (0.45) CYP19A1CYP3A4VNN1
SCHEMBL27287580 0.68 CYP11B1 (0.44) CYP19A1GRM5CYP11B1CYP11B2
SCHEMBL8329925 0.68 KCNJ1 (0.41) CYP19A1GRM5KDM4E
SCHEMBL6063814 0.68 CYP19A1 (0.38) CYP19A1GRM5VNN1CYP11B1CYP11B2
SCHEMBL8328528 0.67 MEN1 (0.49) CYP19A1CYP3A4PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed