SCHEMBL8330253

SCHEMBL8330253

N#Cc1ccc(N(c2ccc(C#N)cc2)c2cncnc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.52
CYP11B2 P19099 3/20 0.39
CYP2A6 P11509 2/20 0.38
ENPP2 Q13822 1/20 0.38
GRM5 P41594 3/20 0.37
ALDH1A1 P00352 2/20 0.37
CA12 O43570 1/20 0.37
CA2 P00918 1/20 0.37
CA3 P07451 1/20 0.37
CA6 P23280 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
TSHR P16473 2/20 0.35
CYP11B1 P15538 2/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324537 0.87 KIF11 (0.53) CYP19A1CYP3A4
SCHEMBL8328528 0.84 MEN1 (0.49) CYP19A1ALDH1A1TSHRCYP3A4CYP2C19
SCHEMBL995812 0.82 CA2 (0.50) CYP2A6ENPP2ALDH1A1CA12CA2
SCHEMBL8329925 0.82 KCNJ1 (0.41) CYP19A1ENPP2GRM5ALDH1A1KDM4E
SCHEMBL8328181 0.79 CYP19A1 (0.38) CYP19A1CYP11B2GRM5CYP11B1CYP3A4
SCHEMBL25543233 0.76 MMP3 (0.56) CYP11B2CYP2A6ENPP2ALDH1A1CA12
SCHEMBL25544161 0.76 MMP3 (0.56) CYP11B2CYP2A6ENPP2ALDH1A1CA12
SCHEMBL8328066 0.75 CYP19A1 (0.44) CYP19A1CYP11B2CYP2A6ALDH1A1CYP11B1
SCHEMBL25543818 0.74 CYP11B2 (0.50) CYP11B2CA12CA2CA9CYP11B1
SCHEMBL25543310 0.74 CYP11B2 (0.50) CYP11B2CA12CA2CA9CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed