SCHEMBL8328239

SCHEMBL8328239

Cc1cc(CCC(C(=O)O)C(=O)O)nc(-n2c(C)ccc2C)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 3/20 0.37
NOS2 P35228 3/20 0.37
NOS3 P29474 2/20 0.37
MYC P01106 5/20 0.35
NR4A1 P22736 3/20 0.33
PTPN7 P35236 3/20 0.33
HSD17B10 Q99714 3/20 0.33
KDM4E B2RXH2 3/20 0.33
MEN1 O00255 3/20 0.33
POLB P06746 3/20 0.33
MAPT P10636 3/20 0.33
KMT2A Q03164 3/20 0.33
TDP1 Q9NUW8 3/20 0.33
CYP2C19 P33261 2/20 0.33
RECQL P46063 2/20 0.33
BLM P54132 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
CYP2C9 P11712 1/20 0.33
APEX1 P27695 2/20 0.33
DHODH Q02127 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329387 0.82 NOS2 (0.55) NOS1NOS2NOS3ESR1
SCHEMBL6767585 0.81 RXRA (0.50) NOS1NOS2NOS3KDM4ERXRA
SCHEMBL6766749 0.80 NOS2 (0.39) NOS1NOS2NOS3PDE10A
SCHEMBL6762802 0.80 CTSB (0.45) MYCNR4A1PTPN7HSD17B10KDM4E
SCHEMBL6164330 0.80 RXRA (0.46) NOS1NOS2NOS3KDM4EMAPT
SCHEMBL5672155 0.79 NOS2 (0.36) NOS1NOS2NOS3
SCHEMBL8326231 0.79 NOS2 (0.41) NOS1NOS2NOS3PDE10A
SCHEMBL8329711 0.79 NOS2 (0.41) NOS1NOS2NOS3PDE10A
SCHEMBL8326237 0.79 NOS2 (0.41) NOS1NOS2NOS3PDE10A
SCHEMBL6765287 0.78 NOS2 (0.38) NOS1NOS2NOS3RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US disclosed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO disclosed