SCHEMBL6762802

SCHEMBL6762802

Cc1cc(CC(=O)O)nc(-n2c(C)ccc2C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSB P07858 3/20 0.45
KLKB1 P03952 2/20 0.45
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 4/20 0.44
POLB P06746 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MYC P01106 7/20 0.38
GAA P10253 3/20 0.37
MAPT P10636 3/20 0.37
NR4A1 P22736 3/20 0.37
AGBL2 Q5U5Z8 1/20 0.36
APEX1 P27695 2/20 0.36
ELANE P08246 2/20 0.36
DUSP3 P51452 2/20 0.36
HPGD P15428 2/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
DHODH Q02127 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6767585 0.82 RXRA (0.50) CTSBKLKB1KDM4ERXRARXRB
SCHEMBL13040659 0.82 KDM4E (0.45) KDM4EALDH1A1POLBTDP1MAPT
SCHEMBL6164330 0.81 RXRA (0.46) KDM4EMAPTRXRARXRBRXRG
SCHEMBL5673102 0.80 NOTUM (0.33) KDM4EALDH1A1POLBL3MBTL1MYC
SCHEMBL8328239 0.80 NOS1 (0.37) CTSBKLKB1KDM4EALDH1A1POLB
SCHEMBL6489717 0.79 CTSB (0.46) CTSBKLKB1KDM4EALDH1A1POLB
SCHEMBL8326929 0.78 NOS2 (0.48) KDM4EALDH1A1L3MBTL1GAAHPGD
SCHEMBL5672155 0.78 NOS2 (0.36)
SCHEMBL2773550 0.77 MYC (0.32) KDM4EALDH1A1L3MBTL1MYCGAA
SCHEMBL5930653 0.77 SMN1; SMN2 (0.36) KDM4EALDH1A1TDP1L3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6762176-B1 INHIBITING NO-SYNTHASE ENZYMES PRODUCING NITROGEN MONOXIDE AND/OR TRAPPING REACTIVE FORMS OF OXYGEN; INHIBIT LIPIDIC PEROXIDATION SOCIETE DE CONSELLS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2004-07-13 US disclosed
US-6727239-B1 INHIBITORY ACTIVITY ON NO- SYNTHASE ENZYMES PRODUCING NITROGEN MONOXIDE NO AND/OR AN ACTIVITY WHICH TRAPS THE REACTIVE OXYGEN SPECIES (ROS) SOCIETE DE CONSEILS DE RECHERCHES ET D'APPLICATIONS SCIENTIFIQUES (S.C.R.A.S.) (FR) 2004-04-27 US disclosed