SCHEMBL8328655

SCHEMBL8328655

Cc1ccc(C2=CC(C)(C)c3ccc(C#Cc4ccccc4C(=O)O)cc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RARB P10826 17/20 0.52
RARA P10276 16/20 0.52
RARG P13631 16/20 0.52
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
HNF4A P41235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5480486 0.85 RARB (0.73) RARBRARARARG
SCHEMBL6240904 0.84 RARB (0.71) RARBRARARARG
SCHEMBL6397552 0.84 RARB (0.51) RARBRARARARG
SCHEMBL8328656 0.80 RARB (0.48) RARBRARARARGNPC1RAB9A
SCHEMBL8772792 0.79 RARB (0.61) RARBRARARARG
SCHEMBL6234600 0.75 RARA (0.53) RARBRARARARG
SCHEMBL8329422 0.73 RARA (0.44) RARBRARARARGNPC1RAB9A
SCHEMBL8335170 0.73 RARB (0.44) RARBRARARARGNPC1RAB9A
SCHEMBL8580705 0.72 RARB (0.65) RARBRARARARGNPC1RAB9A
SCHEMBL8772626 0.72 RARA (0.62) RARBRARARARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958954-A 2,2-DIALKYL-4-ARYL-SUBSTITUTED BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES ALLERGAN SALES, INC. (US) 1999-09-28 US disclosed
US-5952345-A RETINOID ACID RECEPTOR ANTAGONIST; A DERIVATIVES OF ARYL-SUBSTITUTED AND ARYL (3-OXO-1-PROPENLY)-SUBSTITUTED BENZOPYRAN, BENZOTHIOPYRAN, 1,2-DIHYDROQUINOLINE; PREVENTING TOXICITY OR SIDE EFFECTS CAUSED BY RETINOIDS OR VITAMIN A ALLERGAN SALES, INC. (US) 1999-09-14 US disclosed
US-5877207-A SKIN DISORDERS; ANTICARCINOGENIC AGENTS ALLERGAN SALES, INC. (US) 1999-03-02 US disclosed