SCHEMBL8328849

SCHEMBL8328849

O=C(O)c1ccc(F)c(NCCc2cccnc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM6B O15054 1/20 0.50
KDM4C Q9H3R0 1/20 0.50
VNN1 O95497 2/20 0.48
CSNK2A2 P19784 3/20 0.48
CSNK2A1 P68400 3/20 0.48
NAMPT P43490 3/20 0.47
CSNK2B P67870 1/20 0.47
HDAC8 Q9BY41 2/20 0.46
HDAC6 Q9UBN7 2/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC1 Q13547 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
APAF1 O14727 1/20 0.46
PABPC1 P11940 1/20 0.46
CASP6 P55212 1/20 0.46
CASP8 Q14790 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329817 0.83 VNN1 (0.43) KDM6BKDM4CVNN1NAMPTHDAC8
SCHEMBL28679564 0.74 TRPV1 (0.54) KDM6BKDM4CCSNK2A2CSNK2A1NAMPT
SCHEMBL30874169 0.73 ALDH1A1 (0.49) HDAC8HDAC6HDAC1L3MBTL1RAB9A
SCHEMBL10690524 0.73 HCAR3 (0.57) KDM6BKDM4CHDAC8HDAC6HDAC1
SCHEMBL21409362 0.73 ALDH1A1 (0.49) HDAC8HDAC6HDAC1L3MBTL1RAB9A
SCHEMBL6845399 0.72 MRGPRX4 (0.55) KDM4CVNN1
SCHEMBL8996251 0.72 TBXAS1 (0.58) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL5307781 0.71 LTA4H (0.69) L3MBTL1APAF1PABPC1CASP6CASP8
SCHEMBL1116010 0.71 KDM6B (0.59) KDM6BKDM4CHDAC8HDAC6HDAC1
SCHEMBL5353235 0.70 TBXAS1 (0.62) L3MBTL1PTAFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869787-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 1999-03-24 EP disclosed
EP-0869787-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1998-10-14 EP disclosed
WO-1997024119-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed