SCHEMBL8329102

SCHEMBL8329102

O=[N+]([O-])c1ccc(N(Cc2cscn2)c2cncnc2)nc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.38
POLB P06746 2/20 0.37
KMT2A Q03164 5/20 0.34
RAB9A P51151 2/20 0.34
HSP90AA1 P07900 1/20 0.34
CXCR5 P32302 1/20 0.34
APLNR P35414 1/20 0.34
CCR6 P51684 1/20 0.34
GFER P55789 1/20 0.34
CYP1A2 P05177 2/20 0.33
GAA P10253 1/20 0.33
METAP1 P53582 1/20 0.32
MEN1 O00255 3/20 0.32
NPC1 O15118 1/20 0.32
KDM4E B2RXH2 1/20 0.32
AGTR1 P30556 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327951 0.75 SLC29A1 (0.41) PKMPOLBKMT2ARAB9AGAA
SCHEMBL8446530 0.67 CYP19A1 (0.58) KMT2AMETAP1MEN1CYP19A1ALDH1A1
SCHEMBL8327952 0.66 CRHBP (0.47) POLBCYP1A2CYP3A4CYP2C19CYP19A1
SCHEMBL4825951 0.64 LMNA (0.61) KMT2ARAB9AMEN1CYP19A1MAPT
SCHEMBL933269 0.63 PKM (0.57) PKMPOLBKMT2ARAB9AHSP90AA1
SCHEMBL30402495 0.63 PKM (0.57) PKMPOLBKMT2ARAB9AHSP90AA1
SCHEMBL23634077 0.62 PKM (0.74) PKMPOLBKMT2ARAB9AHSP90AA1
SCHEMBL1542306 0.62 PKM (0.54) PKMPOLBKMT2ARAB9AHSP90AA1
SCHEMBL6490056 0.62 ALDH1A1 (0.44) POLBKMT2ARAB9ACYP1A2MEN1
SCHEMBL8327171 0.62 CRHBP (0.42) POLBCYP1A2CYP3A4CYP2C19CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
CN-1039228-C Novel substituted tert-amino compund YAMANOUCHI PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed