SCHEMBL8327951

SCHEMBL8327951

O=[N+]([O-])c1ccc(N(Cc2ccc(F)c(F)c2)c2cncnc2)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC29A1 Q99808 2/20 0.41
PKM P14618 1/20 0.39
MAPT P10636 4/20 0.36
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
POLB P06746 3/20 0.35
CYP3A4 P08684 1/20 0.35
ABCC1 P33527 1/20 0.35
HSPB1 P04792 2/20 0.35
SSTR2 P30874 1/20 0.34
SSTR4 P31391 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
HIF1A Q16665 1/20 0.33
RPS6KB1 P23443 1/20 0.33
AKT1 P31749 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALOX12 P18054 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329102 0.75 PKM (0.38) PKMMAPTALDH1A1NPC1GAA
SCHEMBL8327952 0.73 CRHBP (0.47) ALDH1A1POLBCYP3A4
SCHEMBL8323939 0.72 AR (0.49) NPC1RAB9APOLBHSPB1MEN1
SCHEMBL8327623 0.70 ALDH1A1 (0.50) MAPTALDH1A1NPC1GAARAB9A
SCHEMBL5326091 0.69 MAPT (0.57) SLC29A1MAPTALDH1A1NPC1GAA
SCHEMBL8326188 0.68 CYP19A1 (0.55) MAPTALDH1A1NPC1RAB9APOLB
SCHEMBL8327171 0.68 CRHBP (0.42) MAPTALDH1A1POLBCYP3A4
SCHEMBL8329070 0.68 MMP1 (0.45) MAPTRAB9APOLBIDO1
SCHEMBL8323116 0.67 CYP19A1 (0.39) MAPTPOLBTDP1
SCHEMBL8327043 0.67 CYP19A1 (0.45) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed