SCHEMBL8329362

SCHEMBL8329362

CC(=O)OC[C@H]1O[C@@H](n2cc(F)c(=O)[nH]c2=O)C[C@@H]1OC(C)=O

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
RNASE1 P07998 1/20 0.48
TYMS P04818 1/20 0.46
TK1 P04183 3/20 0.43
ABCG2 Q9UNQ0 3/20 0.42
ABCB1 P08183 1/20 0.42
ESR1 P03372 1/20 0.42
MAPT P10636 1/20 0.42
NT5E P21589 1/20 0.41
P2RY6 Q15077 1/20 0.41
P2RY14 Q15391 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL570200 1.00 LMNA (0.55) LMNASMN1; SMN2RNASE1TYMSTK1
SCHEMBL24595722 0.92 LMNA (0.55) LMNASMN1; SMN2RNASE1TYMSTK1
SCHEMBL6852678 0.89 LMNA (0.67) LMNASMN1; SMN2RNASE1TK1
SCHEMBL16311910 0.89 LMNA (0.57) LMNASMN1; SMN2RNASE1TYMSTK1
SCHEMBL13026818 0.89 LMNA (0.67) LMNASMN1; SMN2RNASE1TK1
SCHEMBL6374113 0.89 LMNA (0.67) LMNASMN1; SMN2RNASE1TK1
SCHEMBL12969271 0.88 RNASE1 (0.61) RNASE1TK1ABCG2ABCB1
SCHEMBL4278968 0.88 RNASE1 (0.61) RNASE1TK1ABCG2ABCB1
SCHEMBL22143532 0.88 RNASE1 (0.61) RNASE1TK1ABCG2ABCB1
SCHEMBL4278972 0.88 RNASE1 (0.61) RNASE1TK1ABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4599404-A BENOYLATION FUNAI PHARMACEUTICAL IND., LTD. (JP) 1986-07-08 US claimed
EP-0009882-A1 2'-Deoxy-5-fluorouridine derivatives, a process for producing the same and antitumor agents comprising the same FUNAI PHARMACEUTICAL IND., LTD. (JP) 1980-04-16 EP claimed
JP-56113795-A None JP disclosed
JP-55035057-A None JP disclosed
US-8916536-B2 Bone-targeting bisphosphonate duplex drugs SCHOTT HERBERT (DE) 2014-12-23 US disclosed
EP-2601202-B1 BONE-TARGETING BISPHOSPHONATE DUPLEX DRUGS SCHOTT HERBERT (DE) 2014-09-03 EP disclosed
US-20130237494-A1 BONE-TARGETING BISPHOSPHONATE DUPLEX DRUGS SCHOTT HERBERT (DE) 2013-09-12 US disclosed
US-5869464-A HAVING LOW TOXICITY, SUSTAINING LOW CONCENTRATION IN BLOOD FOR EXTENDED PERIOD TAIHO PHARMACEUTICAL CO. LTD. (JP) 1999-02-09 US disclosed
EP-0686641-B1 2'-DEOXY-5-FLUOROURIDINE DERIVATIVE, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PROCESS FOR PRODUCING THE SAME, AND ANTITUMOR DRUG TAIHO PHARMACEUTICAL CO LTD (JP) 1998-08-26 EP disclosed
EP-0686641-A1 2'-DEOXY-5-FLUOROURIDINE DERIVATIVE, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PROCESS FOR PRODUCING THE SAME, AND ANTITUMOR DRUG TAIHO PHARMACEUTICAL CO., LTD. (JP) 1995-12-13 EP disclosed
US-4599404-A BENOYLATION FUNAI PHARMACEUTICAL IND., LTD. (JP) 1986-07-08 US disclosed
US-4503045-A ORAL ADMINISTRATION FUNAI YAKUHIN KOGYO KABUSHIKI KAISHA (JP) 1985-03-05 US disclosed
US-4490366-A 2'-Deoxy-5-fluorouridine derivative and a process for producing the same and an antitumor agent comprising the same FUNAI PHARMACEUTICAL IND., LTD. (JP) 1984-12-25 US disclosed
US-4425335-A ANTITUMOR FUNAI KAKUHIN KOGYO KABUSHIKI KAISHA (JP) 1984-01-10 US disclosed
US-4416875-A ANTITUMOR AGENTS FUNAI YAKUHIN KOGYO KABUSHIKI KAISHA (JP) 1983-11-22 US disclosed
EP-0009882-B1 2'-DEOXY-5-FLUOROURIDINE DERIVATIVES, A PROCESS FOR PRODUCING THE SAME AND ANTITUMOR AGENTS COMPRISING THE SAME FUNAI PHARMACEUTICAL IND., LTD. (JP) 1982-03-03 EP disclosed
JP-S56113795-A 2'-DEOXY-3',5'-DI-O-ACETYL-5-FLUOROURIDINE DERIVATIVE, ITS PREPARATION AND ANTITUMOR AGENT CONTAINING THE SAME FUNAI CORP 1981-09-07 JP disclosed
EP-0009882-A1 2'-Deoxy-5-fluorouridine derivatives, a process for producing the same and antitumor agents comprising the same FUNAI PHARMACEUTICAL IND., LTD. (JP) 1980-04-16 EP disclosed
JP-S5535057-A 2'-DEOXY-5-FLUOROURIDINE DERIVATIVE, ITS PREPARATION, AND ANTITUMOR AGENT COMPRISING IT FUNAI CORP 1980-03-11 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130237494-A1 BONE-TARGETING BISPHOSPHONATE DUPLEX DRUGS BPGM, MVD, PPIP5K2 LMNA 3664/4885SMN1; SMN2 3596/4885RNASE1 1254/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.