SCHEMBL8330353

SCHEMBL8330353

Cc1cc(CCCCn2c(C)ccc2C)nc(-n2c(C)ccc2C)c1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 12/20 0.38
NOS1 P29475 10/20 0.36
NOS3 P29474 9/20 0.36
PRKCI P41743 1/20 0.35
TLR8 Q9NR97 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330518 0.95 NOS2 (0.40) NOS2NOS1NOS3PRKCI
SCHEMBL6164525 0.84 NOS2 (0.39) NOS2NOS1NOS3TLR8
SCHEMBL6166695 0.84 NOS2 (0.45) NOS2NOS1NOS3
SCHEMBL13040655 0.82 NOS2 (0.38) NOS2NOS1NOS3TLR8
SCHEMBL6167004 0.82 NOS2 (0.38) NOS2NOS1NOS3TLR8
SCHEMBL13040653 0.82 NOS2 (0.55) NOS2NOS1NOS3
SCHEMBL13040656 0.82 NOS2 (0.55) NOS2NOS1NOS3
SCHEMBL8330686 0.81 NOS1 (0.57) NOS2NOS1NOS3
SCHEMBL8328137 0.80 NOS2 (0.51) NOS2NOS1NOS3
SCHEMBL6164330 0.79 RXRA (0.46) NOS2NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US disclosed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO disclosed