SCHEMBL8330686

SCHEMBL8330686

Cc1cc(CCCCc2ccccc2)nc(-n2c(C)ccc2C)c1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.57
NOS2 P35228 4/20 0.57
NOS3 P29474 3/20 0.57
CYP2D6 P10635 1/20 0.39
BACE1 P56817 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330574 0.97 NOS1 (0.61) NOS1NOS2NOS3CYP2D6BACE1
SCHEMBL7737460 0.91 NOS1 (0.49) NOS1NOS2NOS3BACE1
SCHEMBL2836244 0.82 NOS1 (0.59) NOS1NOS2NOS3
SCHEMBL6164525 0.82 NOS2 (0.39) NOS1NOS2NOS3
SCHEMBL13040653 0.81 NOS2 (0.55) NOS1NOS2NOS3
SCHEMBL6167004 0.81 NOS2 (0.38) NOS1NOS2NOS3
SCHEMBL8330353 0.81 NOS2 (0.38) NOS1NOS2NOS3
SCHEMBL13040655 0.81 NOS2 (0.38) NOS1NOS2NOS3
SCHEMBL13040656 0.81 NOS2 (0.55) NOS1NOS2NOS3
SCHEMBL6164330 0.81 RXRA (0.46) NOS1NOS2NOS3KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US disclosed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO disclosed