SCHEMBL8344859

SCHEMBL8344859

CC(=O)Nc1ccc(C2=CCN(C)CC2)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
QDPR P09417 4/20 0.49
MMP2 P08253 1/20 0.42
MMP3 P08254 1/20 0.42
CTSS P25774 1/20 0.40
PLK1 P53350 1/20 0.39
PLK3 Q9H4B4 1/20 0.39
PLK2 Q9NYY3 1/20 0.39
ULK1 O75385 1/20 0.39
WDR5 P61964 1/20 0.38
PIK3CA P42336 1/20 0.38
CPT1A P50416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27195861 0.79 QDPR (0.50) QDPRMMP2MMP3PLK1PLK3
SCHEMBL8345083 0.76 QDPR (0.54) QDPRMMP2MMP3
SCHEMBL8130409 0.71 HTR6 (0.53)
SCHEMBL13483657 0.71 MAPT (0.55) CTSS
SCHEMBL8915112 0.71 QDPR (0.62) QDPR
SCHEMBL24670132 0.71 MAPT (0.41) QDPRMMP2MMP3WDR5
SCHEMBL8346983 0.70 CTSS (0.48) CTSSPIK3CA
SCHEMBL24669373 0.69 SOS1 (0.49) WDR5
SCHEMBL8613848 0.69 QDPR (0.46) QDPR
SCHEMBL8122236 0.68 HTR6 (0.50) QDPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004022534-A1 ARYLGLYCINE DERIVATIVES FOR USE AS GLYCINE TRANSPORT INHIBITORS NPS ALLELIX CORP. (CA) 2004-03-18 WO disclosed