SCHEMBL8369355

SCHEMBL8369355

COC(=O)c1cccc(S(=O)(=O)c2ccccc2)c1N

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.59
ALDH1A1 P00352 4/20 0.57
GAA P10253 4/20 0.57
HPGD P15428 2/20 0.57
PKM P14618 1/20 0.57
CA1 P00915 1/20 0.56
CA2 P00918 1/20 0.56
CA5A P35218 1/20 0.56
CA9 Q16790 1/20 0.56
CFTR P13569 1/20 0.50
HSD17B10 Q99714 1/20 0.50
HTR6 P50406 3/20 0.47
MMP2 P08253 5/20 0.47
MMP9 P14780 5/20 0.47
MMP8 P22894 5/20 0.47
MMP12 P39900 5/20 0.47
MMP13 P45452 5/20 0.47
MMP14 P50281 5/20 0.47
MMP16 P51512 5/20 0.47
NPC1 O15118 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10589344 0.83 HTR6 (0.55) KDM4EALDH1A1GAAHPGDPKM
SCHEMBL589633 0.81 HTR6 (0.53) KDM4EALDH1A1GAAHPGDPKM
SCHEMBL27497618 0.81 CA1 (0.58) KDM4EALDH1A1GAAHPGDCA1
SCHEMBL2895994 0.77 ALDH1A1 (0.67) KDM4EALDH1A1GAAHPGDCA1
SCHEMBL11661242 0.76 CA1 (0.73) KDM4EALDH1A1GAACA1CA2
SCHEMBL27484282 0.75 HTR6 (0.47) KDM4EALDH1A1GAAHPGDPKM
SCHEMBL6342597 0.75 ALOX15 (0.45) KDM4EALDH1A1GAACA1CA2
SCHEMBL3157582 0.75 MMP2 (0.58) KDM4EALDH1A1GAAHPGDPKM
SCHEMBL28762183 0.74 KDM4E (1.00) KDM4EALDH1A1GAAHPGDPKM
SCHEMBL31634613 0.74 ALDH1A1 (0.58) KDM4EALDH1A1GAAHPGDCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831800-A4 ARYLSULFONYLAMINOBENZENE DERIVATIVES AND THE USE THEREOF AS FACTOR Xa INHIBITORS DIMENSIONAL PHARM INC (US) 1999-03-10 EP disclosed
EP-0831800-A1 ARYLSULFONYLAMINOBENZENE DERIVATIVES AND THE USE THEREOF AS FACTOR Xa INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1998-04-01 EP disclosed
WO-1996040100-A1 ARYLSULFONYLAMINOBENZENE DERIVATIVES AND THE USE THEREOF AS FACTOR Xa INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1996-12-19 WO disclosed