SCHEMBL8377231

SCHEMBL8377231

COCCOc1c(C(ON)C(=O)OC(c2ccccc2)c2ccccc2)cc(OC)c(C#N)c1OCCOC

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
ALDH1A1 P00352 3/20 0.33
HTR1A P08908 2/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
ADRA1B P35368 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPK8 P45983 2/20 0.33
MAPK9 P45984 2/20 0.33
MAPK10 P53779 2/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33
KIF11 P52732 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8378504 0.78 ALDH1A1 (0.34) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8380298 0.77 HTR1A (0.34) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8377229 0.76 KIF11 (0.32) KIF11
SCHEMBL8377243 0.73 TNFRSF1A (0.38) ALDH1A1HSD17B10MAPK8MAPK9MAPK10
SCHEMBL8379339 0.73 HTR1A (0.36) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8636164 0.72 LMNA (0.39) IDO1TDO2ALDH1A1HTR1AADRA1D
SCHEMBL8378913 0.71 ALDH1A1 (0.39) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8377093 0.71 SLC6A5 (0.37) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL8377272 0.70 HTR1A (0.34) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL9065459 0.69 KIF11 (0.33) IDO1TDO2KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883248-A QUATERNARY AMMONIUM INTERMEDIATES ROUSSEL UCLAF (FR) 1999-03-16 US disclosed
US-5763617-A Cephalosporins ROUSSEL UCLAF (FR) 1998-06-09 US disclosed
US-5712266-A Cephalosporins ROUSSEL UCLAF (FR) 1998-01-27 US disclosed