Bromide

Bromide

SCHEMBL83856

Br.CC(CCCl)(CCCl)NCc1ccccc1

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 1/20 0.35
SIGMAR1 known ✓ Q99720 1/20 0.35
CYP3A4 P08684 3/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ATM Q13315 1/20 0.38
IDO1 P14902 2/20 0.38
THRB P10828 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
RIPK1 Q13546 1/20 0.38
CYP2D6 P10635 2/20 0.37
LMNA P02545 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 2/20 0.36
TAAR1 Q96RJ0 1/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1839087 0.98 CYP3A4 (0.42) CYP3A4MAPTKDM4EATMIDO1
SCHEMBL20686991 0.76 RIPK1 (0.50) CYP3A4MAPTKDM4EATMIDO1
Bromide SCHEMBL11038149 0.76 CYP3A4 (0.50) CYP3A4MAPTKDM4EATMIDO1
SCHEMBL14145021 0.76 CYP3A4 (0.50) CYP3A4MAPTKDM4EATMIDO1
SCHEMBL6132599 0.75 HTT (0.50) CYP3A4MAPTKDM4EATMIDO1
SCHEMBL11751773 0.74 CYP2D6 (0.48) CYP3A4MAPTKDM4EATMIDO1
SCHEMBL928816 0.74 CYP3A4 (0.48) CYP3A4MAPTKDM4EATMIDO1
SCHEMBL125129 0.73 CYP3A4 (0.52) CYP3A4MAPTKDM4EATMIDO1
SCHEMBL9779031 0.73 HTT (0.45) CYP3A4MAPTKDM4EATMIDO1
Hydrochloric Acid SCHEMBL538794 0.71 CYP3A4 (0.56) CYP3A4MAPTKDM4EATMIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1101 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11717481-B2 Reduction of flake-like aggregation in nanoparticulate active agent compositions ALKERMES PHARMA IRELAND LIMITED (IE) 2023-08-08 US claimed
US-20220211626-A1 REDUCTION OF FLAKE-LIKE AGGREGATION IN NANOPARTICULATE ACTIVE AGENT COMPOSITIONS JPMORGAN CHASE BANK, N.A. AS ADMINISTRATIVE AGENT 2022-07-07 US claimed
US-11253478-B2 Reduction of flake-like aggregation in nanoparticulate active agent compositions ALKERMES PHARMA IRELAND LIMITED (IE) 2022-02-22 US claimed
EP-3755148-A1 NANOSUSPENSIONS OF SALSALATE AND METHODS OF USING THE SAME RHNanoPharma (US) 2020-12-30 EP claimed
US-20200390737-A1 NANOSUSPENSIONS OF SALSALATE AND METHODS OF USING THE SAME RHNANOPHARMA (US) 2020-12-17 US claimed
WO-2019165240-A1 NANOSUSPENSIONS OF SALSALATE AND METHODS OF USING THE SAME RHNANOPHARMA (US) 2019-08-29 WO claimed
US-20180250229-A1 REDUCTION OF FLAKE-LIKE AGGREGATION IN NANOPARTICULATE ACTIVE AGENT COMPOSITIONS ALKERMES PHARMA IRELAND LIMITED (IE) 2018-09-06 US claimed
US-9974748-B2 Reduction of flake-like aggregation in nanoparticulate active agent compositions ALKERMES PHARMA IRELAND LIMITED (IE) 2018-05-22 US claimed
US-9974746-B2 Reduction of flake-like aggregation in nanoparticulate active agent compositions ALKERMES PHARMA IRELAND LIMITED (IE) 2018-05-22 US claimed
US-9974747-B2 Reduction of flake-like aggregation in nanoparticulate active agent compositions ALKERMES PHARMA IRELAND LIMITED (IE) 2018-05-22 US claimed
WO-2003080024-A2 NANOPARTICULATE COMPOSITIONS OF MAP KINASE INHIBITORS ELAN PHARMA INTERNATIONAL, LTD. (IE) 2003-10-02 WO claimed
WO-2003080023-A2 FAST DISSOLVING DOSAGE FORMS HAVING REDUCED FRIABILITY ELAN PHARMA INTERNATIONAL LIMITED (IE) 2003-10-02 WO claimed
WO-2003080027-A1 NANOPARTICULATE COMPOSITIONS OF ANGIOGENESIS INHIBITORS ELAN PHARMA INTERNATIONAL, LTD. (IE) 2003-10-02 WO claimed
US-20030185869-A1 Having lysozyme adsorbed onto or associated with the surface of an active agent ELAN PHARMA INTERNATIONAL LTD. 2003-10-02 US claimed
US-20030181411-A1 Contacting and adsorbing an insoluble enzyme inhibitor with a surface stabilizer ELAN PHARMA INTERNATIONAL LTD. 2003-09-25 US claimed
WO-2003066021-A2 DRUG NANOPARTICLES WITH LYSOZYME SURFACE STABILISER ELAN PHARMA INTERNATIONAL, LTD. (IE) 2003-08-14 WO claimed
US-20030137067-A1 Compositions having a combination of immediate release and controlled release characteristics ELAN PHARMA INTERNATIONAL LTD. 2003-07-24 US claimed
US-20030095928-A1 Nanoparticulate insulin ELAN PHARMA INTERNATIONAL LIMITED 2003-05-22 US claimed
WO-2003030872-A2 COMPOSITIONS HAVING A COMBINATION OF PARTICLES FOR IMMEDIATE RELEASE AND FOR CONTROLLED RELEASE ELAN PHARMA INTERNATIONAL LTD. (IE) 2003-04-17 WO claimed
WO-2003024425-A1 NANOPARTICULATE INSULIN FORMULATIONS ELAN PHARMA INTERNATIONAL, LTD. (IE) 2003-03-27 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200390737-A1 NANOSUSPENSIONS OF SALSALATE AND METHODS OF USING THE SAME TUBAL3, TUBB6, TUBA1A SLC6A2 825/4885SIGMAR1 1253/4885CYP3A4 1404/4885
US-20030181411-A1 Contacting and adsorbing an insoluble enzyme inhibitor with a surface stabilizer PACSIN2, MAP3K20, MAP3K2 SLC6A2 2874/4885SIGMAR1 2060/4885CYP3A4 3419/4885
US-20030137067-A1 Compositions having a combination of immediate release and controlled release characteristics NAPA, CD63, RPL36 SLC6A2 773/4885SIGMAR1 259/4885CYP3A4 2022/4885
US-20030185869-A1 Having lysozyme adsorbed onto or associated with the surface of an active agent LPO, LCT, CTSA SLC6A2 2817/4885SIGMAR1 1877/4885CYP3A4 1457/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.