SCHEMBL8399072

SCHEMBL8399072

CCCCc1ccccc1OCc1ccccc1N(CC)C(=O)C=NOC

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
PPARD Q03181 1/20 0.36
CYP3A4 P08684 3/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTGER1 P34995 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGER3 P43115 1/20 0.35
PTGER2 P43116 1/20 0.35
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
ABCB1 P08183 1/20 0.34
PPARA Q07869 1/20 0.34
LTB4R Q15722 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
LMNA P02545 1/20 0.34
SNCA P37840 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399032 0.97 THRA (0.45) THRATHRBPPARDCYP3A4CYP1A2
SCHEMBL8396234 0.94 PPARD (0.39) THRATHRBPPARDCYP3A4BCHE
SCHEMBL8398724 0.91 NISCH (0.38) THRBCYP3A4LMNASNCA
SCHEMBL8400210 0.88 THRA (0.41) THRATHRBPPARDCYP3A4CYP1A2
SCHEMBL8395408 0.86 CYP3A4 (0.43) CYP3A4LMNA
SCHEMBL8397742 0.85 THRA (0.46) THRATHRBPPARDPTGER1PTGER4
SCHEMBL8399060 0.85 TP53 (0.45) THRBLTB4RLTB4R2LMNA
SCHEMBL8399129 0.85 LMNA (0.41) THRBCYP3A4LTB4RLTB4R2LMNA
SCHEMBL8519936 0.83 NISCH (0.36) CYP3A4CYP1A2CYP2C19PPARALMNA
SCHEMBL8395164 0.83 CYP3A4 (0.41) CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0644183-B1 Process of producing N-alkylacetamides SHIONOGI & CO (JP) 1999-06-02 EP disclosed
US-5498792-A Process of producing N-alkylacetamides SHIONOGI & CO., LTD. (JP) 1996-03-12 US disclosed
EP-0644183-A2 Process of producing N-alkylacetamides SHIONOGI & CO., LTD. (JP) 1995-03-22 EP disclosed