SCHEMBL8400189

SCHEMBL8400189

CCCc1cccc(NCc2nc3cc(F)cc(F)c3s2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 6/20 0.36
NOS1 P29475 4/20 0.34
NOS2 P35228 3/20 0.34
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
NPR1 P16066 1/20 0.32
S1PR4 O95977 1/20 0.32
S1PR5 Q9H228 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399113 0.85 NOS1 (0.44) AKR1B1NOS1
SCHEMBL8396076 0.84 MEN1 (0.34) NOS1NOS2GRIN2DGRIN3BGRIN1
SCHEMBL8396047 0.82 AKR1B1 (0.39) AKR1B1
SCHEMBL8399351 0.82 AKR1B1 (0.46) AKR1B1NOS1
SCHEMBL8399732 0.81 AKR1B1 (0.42) AKR1B1
SCHEMBL8399092 0.81 AKR1B1 (0.38) AKR1B1NOS1
SCHEMBL8399257 0.81 SYK (0.44) AKR1B1HDAC4MEF2D
SCHEMBL8399287 0.79 AKR1B1 (0.35) AKR1B1
SCHEMBL8395489 0.78 AKR1B1 (0.39) AKR1B1
SCHEMBL8399262 0.77 AKR1B1 (0.40) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed