SCHEMBL8401465

SCHEMBL8401465

CCOc1c(-n2c(CC)nc3ccccc3c2=O)cccc1[N+](=O)[O-]

nearest known ligand 0.76

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.76
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
LMNA P02545 2/20 0.60
MAPT P10636 2/20 0.60
GAA P10253 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.56
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
HIF1A Q16665 6/20 0.48
POLB P06746 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8403511 0.81 L3MBTL1 (0.58) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8399362 0.80 ALDH1A1 (0.47) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4465299 0.79 L3MBTL1 (0.79) ALDH1A1LMNAL3MBTL1HIF1A
SCHEMBL1592847 0.75 ALDH1A1 (0.57) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11435540 0.74 L3MBTL1 (0.71) ALDH1A1LMNAMAPTGAAL3MBTL1
SCHEMBL14305182 0.71 L3MBTL1 (0.67) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8402756 0.71 ALDH1A1 (0.55) ALDH1A1LMNAMAPTL3MBTL1MEN1
SCHEMBL14304598 0.71 L3MBTL1 (0.70) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8242227 0.70 NPC1 (0.70) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL14303441 0.70 HIF1A (0.68) ALDH1A1LMNAL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5885997-A Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-03-23 US disclosed