SCHEMBL8414721

SCHEMBL8414721

COC(=O)C(CC(=O)OC(C)(C)C)NC(=O)C(NC(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.52
CTSD P07339 2/20 0.49
CTSK P43235 4/20 0.48
KYNU Q16719 1/20 0.48
SYK P43405 1/20 0.48
CTSB P07858 2/20 0.48
KLK5 Q9Y337 1/20 0.48
REN P00797 1/20 0.47
CA2 P00918 1/20 0.47
CA5A P35218 1/20 0.47
CTSL P07711 2/20 0.47
CTSS P25774 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8411381 0.91 CASP3 (0.55) CASP3CTSDCTSKCTSBREN
SCHEMBL19694834 0.89 KYNU (0.56) CTSKKYNUSYKCTSBKLK5
SCHEMBL19694832 0.89 KYNU (0.56) CTSKKYNUSYKCTSBKLK5
SCHEMBL4256075 0.89 KYNU (0.56) CTSKKYNUSYKCTSBKLK5
SCHEMBL626800 0.89 CASP3 (0.49) CASP3CTSDCTSKSYKCTSB
SCHEMBL4422741 0.89 CASP3 (0.49) CASP3CTSDCTSKSYKCTSB
SCHEMBL10074125 0.89 CASP3 (0.49) CASP3CTSDCTSKSYKCTSB
SCHEMBL14190228 0.85 CTSL (0.61) CTSKKYNUSYKCTSBKLK5
SCHEMBL5493054 0.84 CASP3 (0.58) CASP3CTSDSYKCTSBCA2
SCHEMBL7303642 0.84 CTSK (0.56) CASP3CTSKSYKCTSBREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0932598-A1 ASPARTATE ESTER INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1999-08-04 EP disclosed
WO-1998016502-A1 ASPARTATE ESTER INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME WARNER-LAMBERT COMPANY (US) 1998-04-23 WO disclosed