SCHEMBL8420103

SCHEMBL8420103

O=S(=O)(Nn1nc(-c2cccc(Cl)c2)cc1-c1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.45
KAT6A Q92794 2/20 0.45
PGR P06401 2/20 0.44
NAT1 P18440 1/20 0.42
KDM1A O60341 6/20 0.41
MAOA P21397 3/20 0.41
AURKA O14965 1/20 0.41
MALT1 Q9UDY8 3/20 0.41
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
PPP1CA P62136 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8422269 0.95 PGR (0.44) PTGS2KAT6APGRNAT1KDM1A
SCHEMBL8641119 0.93 AURKA (0.46) PTGS2KAT6AKDM1AMAOAAURKA
SCHEMBL8421776 0.92 KDM1A (0.47) PTGS2KAT6ANAT1KDM1AMAOA
SCHEMBL8420734 0.90 MALT1 (0.43) KAT6APGRKDM1AMAOAAURKA
SCHEMBL8423597 0.90 KAT6A (0.42) PTGS2KAT6AKDM1AMAOAAURKA
SCHEMBL8421734 0.90 KDM1A (0.43) KAT6APGRKDM1AMAOAAURKA
SCHEMBL8424142 0.90 KAT6A (0.47) KAT6APGRKDM1AMAOAAURKA
SCHEMBL8422282 0.90 KDM1A (0.43) PTGS2KAT6AKDM1AMAOAAURKA
SCHEMBL8420836 0.88 KMO (0.49) PTGS2KAT6APGRNAT1KDM1A
SCHEMBL8419964 0.88 MAPT (0.42) PTGS2KAT6APGRKDM1AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed