SCHEMBL8428958

SCHEMBL8428958

COc1cc2[nH]c(S)nc2cc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 10/20 0.37
ILK Q13418 1/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
EHMT2 Q96KQ7 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PDE10A Q9Y233 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211457 0.86 AMY1A (0.45) AMY1AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9455942 0.81 AMY1A (0.47) AMY1AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL10834064 0.80 PGK1 (0.46) AMY1AALDH1A1EGLN1
SCHEMBL213270 0.80 KDM4E (0.49) KDM4EALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL9531757 0.78 ATP4A (0.48) AMY1AGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL210918 0.77 ACHE (0.39) KDM4EEGLN1
SCHEMBL10834070 0.77 EGLN1 (0.47) AMY1AEGLN1
SCHEMBL15647865 0.76 GRIN2D (0.47) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9528285 0.74 ATP4A (0.43) AMY1AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL14502996 0.74 MEN1 (0.43) AMY1AKDM4EALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922720-A PHARMACEUTICAL FOR USE IN TREATMENT OF DISEASES BASED ON HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1999-07-13 US disclosed
EP-0772611-A1 PIPERAZINE THIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1997-05-14 EP disclosed
WO-1996002534-A1 PIPERAZINE THIOPYRIDINES FOR CONTROLLING HELICOBACTER BACTERIA BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1996-02-01 WO disclosed