SCHEMBL7375074

SCHEMBL7375074

CC(C)COC(=O)N(NC(=O)c1cc(NC(=N)N)cc(C(F)(F)F)c1)C(Cc1ccccc1)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 5/20 0.38
RHOC P08134 1/20 0.36
RHOA P61586 1/20 0.36
P2RX1 P51575 1/20 0.36
BCHE P06276 1/20 0.35
NNMT P40261 1/20 0.35
CYP1A2 P05177 2/20 0.35
UBE2M P61081 3/20 0.34
DCUN1D1 Q96GG9 3/20 0.34
USP2 O75604 2/20 0.34
CYP3A4 P08684 2/20 0.34
NR1I2 O75469 1/20 0.34
ADRB1 P08588 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
CHRM3 P20309 1/20 0.34
SLC6A2 P23975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7375612 1.00 TRPA1 (0.38) TRPA1RHOCRHOAP2RX1BCHE
SCHEMBL7382269 0.87 NR1H4 (0.41)
SCHEMBL7375082 0.86 NNMT (0.34) TRPA1RHOCRHOABCHENNMT
SCHEMBL7375079 0.86 NNMT (0.34) TRPA1RHOCRHOABCHENNMT
SCHEMBL8429038 0.79 TACR1 (0.34) TRPA1CYP1A2UBE2MDCUN1D1USP2
SCHEMBL7375077 0.79 RHOC (0.39) TRPA1RHOCRHOAP2RX1CYP1A2
SCHEMBL7409600 0.78 MAPT (0.42)
SCHEMBL7375593 0.77 ALDH1A1 (0.42)
SCHEMBL7466483 0.76 NPC1 (0.45)
SCHEMBL7378843 0.75 ITGB1 (0.47) P2RX1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP claimed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO claimed