SCHEMBL8435374

SCHEMBL8435374

C=CCOc1cc2ccc(-c3ccc(O)cn3)cc2c(F)n1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.35
MAPT P10636 1/20 0.34
TDO2 P48775 1/20 0.33
ESR1 P03372 3/20 0.32
ESR2 Q92731 3/20 0.32
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
ALDH2 P05091 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
SQOR Q9Y6N5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8437979 0.86 MAPT (0.38) HIF1AMAPTESR1ESR2ALDH2
SCHEMBL8299691 0.80 RAB9A (0.44) MAPTTDO2ESR1ESR2ALDH2
SCHEMBL9618499 0.72 MAPT (0.46) MAPTALDH2MAOAMAOBMGAM
SCHEMBL8427259 0.69 MAPT (0.40) HIF1AMAPT
SCHEMBL9618725 0.67 GAA (0.44) MAPTALDH2MAOAMAOBMGAM
SCHEMBL8437415 0.66 GABRA1 (0.42) MAPTESR1ESR2ALDH2GAA
SCHEMBL8423689 0.65 MAPT (0.30) MAPT
SCHEMBL8440460 0.65 MAPT (0.30) HIF1AMAPT
SCHEMBL9449606 0.64 CYP11B1 (0.39) MAPTESR1ESR2HSD17B1HSD17B2
SCHEMBL9278177 0.63 SMN1; SMN2 (0.50) MAPTHSD17B1HSD17B2ALDH2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825987-B1 1-FLUORISOQUINOLINE DERIVATIVES AND THE USE THEREOF IN LIQUID CRYSTALLINE MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 1999-12-01 EP disclosed
EP-0824522-B1 1,8-DIFLUORISOQUINOLINE DERIVATIVES AND THE USE THEREOF IN LIQUID CRYSTALLINE MIXTURES AVENTIS RES & TECH GMBH & CO (DE) 1999-10-27 EP disclosed
US-5911913-A 1-fluoroisoquinoline derivatives and the use thereof in liquid crystalline mixtures HOECHST AKTIENGESELLSCHAFT (DE) 1999-06-15 US disclosed
US-5882546-A 1,8-Difluorisoquinoline derivatives and the use thereof in liquid crystalline mixtures HOECHST AKTIENGESELLSCHAFT (DE) 1999-03-16 US disclosed