SCHEMBL845442

SCHEMBL845442

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)c3ncccc3O)cc2)cc1)[C@@H]1CCCN1C(=O)c1ncccc1O

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 1/20 0.43
RHOC P08134 1/20 0.42
RHOA P61586 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
PABPC1 P11940 1/20 0.42
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.41
MAPK1 P28482 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845697 0.89 ALDH1A1 (0.45) CYP2C9CYP2C19MAPTRHOCRHOA
SCHEMBL13272509 0.86 TRPV1 (0.45) CYP2C9CYP2C19TRPV1PABPC1ALDH1A1
SCHEMBL845841 0.86 TRPV1 (0.45) CYP2C9CYP2C19TRPV1PABPC1ALDH1A1
SCHEMBL845651 0.84 CYP2C9 (0.43) CYP2C9CYP2C19RHOCRHOATRPV1
SCHEMBL845699 0.84 RHOC (0.48) RHOCRHOAHTT
SCHEMBL845048 0.83 DGAT1 (0.50) CYP2C9CYP2C19MAPTRHOCRHOA
SCHEMBL845330 0.83 GAA (0.47) CYP2C9CYP2C19PABPC1ALDH1A1HTT
SCHEMBL845501 0.83 HCRTR1 (0.47) CYP2C9CYP2C19MAPTRHOCRHOA
SCHEMBL845708 0.82 RHOC (0.46) CYP2C9CYP2C19MAPTRHOCRHOA
SCHEMBL844980 0.82 ALDH1A1 (0.45) CYP2C9CYP2C19MAPTRHOCRHOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
EP-1893573-B1 INHIBITORS OF HCV REPLICATION BRISTOL MYERS SQUIBB CO (US) 2010-07-21 EP disclosed