SCHEMBL8458372

SCHEMBL8458372

CCN1CCNCC1c1ccc(F)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 9/20 0.39
HTR2C P28335 2/20 0.38
HTR2A P28223 1/20 0.38
HTR2B P41595 1/20 0.38
KDM1A O60341 1/20 0.36
MAOB P27338 1/20 0.36
AKT2 P31751 3/20 0.35
SGK1 O00141 2/20 0.34
RPS6KB1 P23443 2/20 0.34
PRKCQ Q04759 2/20 0.34
ROCK1 Q13464 2/20 0.34
RPS6KA1 Q15418 2/20 0.34
AKT3 Q9Y243 2/20 0.34
ROCK2 O75116 1/20 0.34
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30853839 0.82 HTR3A (0.44) HTR2CHTR2AHTR2B
SCHEMBL22382688 0.81 RIPK1 (0.43) HTR2CHTR2AHTR2BKDM1AMAOB
SCHEMBL18741430 0.80 ADRB1 (0.40) HTR2CHTR2AHTR2BKDM1AALDH1A1
SCHEMBL5240098 0.79 PDE4B (0.43) HTR2CHTR2AHTR2BALDH1A1TSHR
SCHEMBL410563 0.78 P2RX7 (0.43) HTR2CHTR2AHTR2B
SCHEMBL470870 0.78 P2RX7 (0.43) HTR2CHTR2AHTR2B
SCHEMBL18950390 0.78 HTR2C (0.46) HTR2CHTR2AHTR2BKDM1A
SCHEMBL8588169 0.75 HTR2C (0.46) HTR2CHTR2AHTR2BKDM1AMAOB
SCHEMBL7584443 0.74 TDP1 (0.40) HTR2CHTR2AHTR2BL3MBTL1
SCHEMBL7582143 0.73 CHRM3 (0.41) HTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925302-A1 PALLADIUM CATALYZED INDOLIZATION Merck & Co., Inc. (US) 1999-06-30 EP claimed
WO-1998006725-A1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO., INC. (US) 1998-02-19 WO claimed