SCHEMBL8465748

SCHEMBL8465748

C=C(C)C(=O)Nc1ccc(Nc2ccc(OC)cc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.58
RAB9A P51151 5/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
MAPT P10636 4/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
KDM4E B2RXH2 2/20 0.57
GAA P10253 2/20 0.57
THRB P10828 1/20 0.57
MAPK1 P28482 1/20 0.57
RECQL P46063 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
TGM2 P21980 1/20 0.54
RXFP1 Q9HBX9 1/20 0.54
TP53 P04637 1/20 0.53
ALOX15 P16050 1/20 0.53
POLB P06746 1/20 0.51
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51
CYP19A1 P11511 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5005383 0.95 NPC1 (0.63) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL13609815 0.86 SMN1; SMN2 (0.56) NPC1RAB9ASMN1; SMN2MAPTTHRB
SCHEMBL11299833 0.83 MEN1 (0.59) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL8467758 0.83 LMNA (0.64) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL9571811 0.82 MTNR1A (0.71) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL6396790 0.82 RAB9A (0.76) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL439393 0.82 RXFP1 (0.74) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL9095411 0.81 KMT2A (0.63) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1
SCHEMBL166821 0.81 MAPT (0.67) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL8465247 0.81 RXFP1 (0.59) NPC1RAB9ASMN1; SMN2MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5936038-A MIXTURE CONTAINING ELASTOMER HAVING PENDANT REACTIVE AMINE GROUP AND PHENOLIC RESIN CURATIVE THE UNIVERSITY OF AKRON (US) 1999-08-10 US claimed
US-5936038-A MIXTURE CONTAINING ELASTOMER HAVING PENDANT REACTIVE AMINE GROUP AND PHENOLIC RESIN CURATIVE THE UNIVERSITY OF AKRON (US) 1999-08-10 US disclosed
EP-0570825-B1 Tire sidewall composition containing silica having low PH GOODYEAR TIRE & RUBBER (US) 1996-08-07 EP disclosed
EP-0475215-B1 Carboxylic acid esters with thio groups GOODYEAR TIRE & RUBBER (US) 1994-10-19 EP disclosed
EP-0570825-A1 Tire sidewall composition containing silica having low PH THE GOODYEAR TIRE & RUBBER COMPANY (US) 1993-11-24 EP disclosed
US-5244028-A Natural rubber or polybutadiene, silica, antidegradation agent, carbon black THE GOODYEAR TIRE & RUBBER COMPANY (US) 1993-09-14 US disclosed
US-5216049-A A phenolic or amine stabilizer and an organothioalkylene styrene bound to a polymer; aging resistance; rubbers THE GOODYEAR TIRE & RUBBER COMPANY (US) 1993-06-01 US disclosed
EP-0475215-A1 Carboxylic acid esters with thio groups THE GOODYEAR TIRE & RUBBER COMPANY (US) 1992-03-18 EP disclosed
US-5069819-A SYNERGISTS FOR CONVENTIONAL PHENOLIC AND AMINE ANTIOXIDANTS THE GOODYEAR TIRE & RUBBER COMPANY (US) 1991-12-03 US disclosed
US-4281080-A TACKIFIERS FOR RUBBERS THE GOODYEAR TIRE & RUBBER COMPANY (US) 1981-07-28 US disclosed
US-4010140-A Age resistant resin compositions and admixtures useful as adhesives THE GOODYEAR TIRE & RUBBER COMPANY (US) 1977-03-01 US disclosed