SCHEMBL8469856

SCHEMBL8469856

CCC(c1cccc2c1C(=O)NC2=O)N1CCC(c2noc3cc(F)ccc23)CC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.51
SLC6A4 P31645 1/20 0.51
HTR2A P28223 14/20 0.48
HTR2C P28335 6/20 0.48
ACHE P22303 2/20 0.47
HTR7 P34969 7/20 0.46
KCNH2 Q12809 7/20 0.46
HTR1A P08908 2/20 0.46
DRD1 P21728 1/20 0.44
DRD3 P35462 1/20 0.44
HTR6 P50406 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664540 0.94 DRD2 (0.52) DRD2SLC6A4HTR2AHTR2CACHE
SCHEMBL8352941 0.89 DRD2 (0.48) DRD2SLC6A4HTR2AHTR2CACHE
SCHEMBL1545276 0.79 ACHE (0.59) DRD2SLC6A4HTR2AHTR2CACHE
SCHEMBL8469854 0.77 ACHE (0.57) DRD2SLC6A4HTR2AACHEHTR1A
SCHEMBL7744954 0.77 DRD2 (0.52) DRD2SLC6A4HTR2AHTR2CACHE
SCHEMBL8345682 0.77 HTR2C (0.57) DRD2SLC6A4HTR2AHTR2CACHE
SCHEMBL8648906 0.77 DRD2 (0.51) DRD2SLC6A4HTR2AHTR2CACHE
SCHEMBL8664537 0.77 DRD2 (0.57) DRD2SLC6A4HTR2AACHEHTR6
Hydrochloric Acid SCHEMBL8463604 0.76 HTR2C (0.56) DRD2SLC6A4HTR2AHTR2CACHE
SCHEMBL8347635 0.76 DRD2 (0.54) DRD2SLC6A4HTR2AHTR2CACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889035-A 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. (US) 1999-03-30 US disclosed
US-5874435-A PSYCHOLOGICAL DISORDERS; ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1999-02-23 US disclosed
US-5854243-A 3-heteroaryl-1-pyrrolidinealkylthiols and derivatives thereof and their therapeutic utility HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1998-12-29 US disclosed
US-5843977-A (3-heteroaryl-1-pyrrolidinyl) alkoxy!-3,4-dihydro-1(2H)-naphthalenones and related compounds and their therapeutic utility HOECHST MARION ROSUEEL, INC. 1998-12-01 US disclosed
US-5811435-A 2- (4-heteroaryl-1-piperidinyl)alkyl!-1,3-dioxanes and related compounds and their therapeutic utility HOECHST MARION RUSSEL, INC. 1998-09-22 US disclosed