SCHEMBL8485672

SCHEMBL8485672

O=NOC(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.55
KMT2A Q03164 5/20 0.54
MEN1 O00255 3/20 0.54
ADRA2A P08913 2/20 0.54
MAPK1 P28482 2/20 0.54
LMNA P02545 1/20 0.54
CYP3A4 P08684 1/20 0.54
HTR1A P08908 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
ADRA2B P18089 1/20 0.54
ADRA2C P18825 1/20 0.54
MAOA P21397 1/20 0.54
ADRA1D P25100 1/20 0.54
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
CYP2C19 P33261 1/20 0.54
ADRA1A P35348 1/20 0.54
DRD3 P35462 1/20 0.54
OPRK1 P41145 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28626254 0.78 HTT (0.38) AKR1B1KMT2AMEN1ADRA2AMAPK1
SCHEMBL3743731 0.77 AKR1B1 (0.59) AKR1B1KMT2AMEN1ADRA2AMAPK1
SCHEMBL28634747 0.75 P2RX7 (0.38) KMT2AMEN1LMNACYP3A4MAPT
SCHEMBL13739934 0.75 KMT2A (0.65) AKR1B1KMT2AMEN1ADRA2AMAPK1
SCHEMBL1429298 0.74 AKR1B1 (0.55) AKR1B1KMT2AMEN1ADRA2AMAPK1
SCHEMBL1395814 0.74 AKR1B1 (0.65) AKR1B1KMT2AMEN1ADRA2AMAPK1
Ammonia Solution, Strong SCHEMBL27532390 0.73 AKR1B1 (0.53) AKR1B1KMT2AMEN1ADRA2AMAPK1
Hydrochloric Acid SCHEMBL5297667 0.72 ADRA2A (0.65) AKR1B1KMT2AMEN1ADRA2AMAPK1
SCHEMBL4102194 0.72 LMNA (0.59) KMT2AMEN1LMNACYP3A4CYP2D6
SCHEMBL2525484 0.71 AKR1B1 (0.68) AKR1B1KMT2AMEN1ADRA2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962492-A ANTIASTHMA AGENTS; ANTIINFLAMMATORY AGENTS CELLTECH THERAPEUTICS LIMITED (GB) 1999-10-05 US disclosed