SCHEMBL8488203

SCHEMBL8488203

CNC(CON1C(=O)SC(Cc2ccccc2)C1=O)CC1c2c(C)c(O)c(C)c(C)c2OC1(C)C

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8487799 0.89 KDM4E (0.33) KDM4EMAPT
SCHEMBL8487391 0.79 ALOX5 (0.41) MAPTPPARG
SCHEMBL8486948 0.75 MAPT (0.44) KDM4EMAPTPPARG
SCHEMBL8484773 0.71 MAPT (0.33) KDM4EMAPTPPARG
SCHEMBL8487346 0.70 PSEN1 (0.36) KDM4EMAPTPPARG
SCHEMBL6032172 0.65 MAPT (0.53) KDM4EMAPTPPARG
SCHEMBL8857258 0.63 KDM4E (0.40) KDM4EMAPTPPARG
SCHEMBL8484201 0.62 SIGMAR1 (0.45) KDM4EMAPT
SCHEMBL7469293 0.62 MAPT (0.56) KDM4EMAPTPPARG
SCHEMBL8523887 0.62 MAPT (0.43) KDM4EMAPTPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925656-A CONTAINING A 2,4-DIOXOTRIAZOLIDINE RING DR. REDDY'S RESEARCH FOUNDATION (IN) 1999-07-20 US disclosed