SCHEMBL8499012

SCHEMBL8499012

C=CCC(=O)Oc1ccc(Oc2c(-c3ccc(OC)c(Cl)c3)ccc3ccccc23)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 7/20 0.40
ERN1 O75460 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTGS2 P35354 3/20 0.37
POLB P06746 1/20 0.36
PTGS1 P23219 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAOB P27338 1/20 0.36
STK39 Q9UEW8 1/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
GLO1 Q04760 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8500218 0.88 THRA (0.36) TDP1L3MBTL1ALDH1A1ESR1ESR2
SCHEMBL8501370 0.86 L3MBTL1 (0.48) NPBWR1TDP1L3MBTL1KDM4EALDH1A1
SCHEMBL8499017 0.83 AKR1C3 (0.39) NPBWR1ERN1PTGS2PTGS1KDM4E
SCHEMBL8496759 0.81 ALDH1A1 (0.39) NPBWR1ERN1PTGS2PTGS1KDM4E
SCHEMBL8500428 0.81 ESR1 (0.41) TDP1L3MBTL1ALDH1A1ESR1ESR2
SCHEMBL7184010 0.81 ESR1 (0.43) NPBWR1ERN1PTGS2KDM4EALDH1A1
SCHEMBL7184005 0.81 ESR1 (0.43) NPBWR1ERN1PTGS2KDM4EALDH1A1
SCHEMBL7182545 0.80 ESR1 (0.52) KDM4EALDH1A1ESR1ESR2
SCHEMBL7182554 0.80 ESR1 (0.52) KDM4EALDH1A1ESR1ESR2
SCHEMBL7935041 0.80 ADORA2A (0.45) NPBWR1ERN1PTGS2PTGS1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed