SCHEMBL8511121

SCHEMBL8511121

CC(C)(C)c1cc(-c2ccnc(N3CCNCC3)n2)ccc1OC1CCCC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMO O15229 4/20 0.46
DKK1 O94907 3/20 0.41
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
ROCK2 O75116 2/20 0.40
ADRB1 P08588 1/20 0.39
MYLK4 Q86YV6 2/20 0.38
STK17A Q9UEE5 2/20 0.38
PRKD1 Q15139 2/20 0.38
PRKD2 Q9BZL6 2/20 0.38
CLK4 Q9HAZ1 1/20 0.37
TBK1 Q9UHD2 1/20 0.37
PDE4D Q08499 2/20 0.37
TLR9 Q9NR96 1/20 0.37
TLR7 Q9NYK1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8533322 0.99 KMO (0.46) KMODKK1CTSSCTSKROCK2
SCHEMBL8514330 0.88 DKK1 (0.55) KMODKK1ROCK2
Hydrochloric Acid SCHEMBL8510232 0.87 DKK1 (0.54) KMODKK1ROCK2
SCHEMBL8511790 0.83 ROCK2 (0.41) KMODKK1ROCK2ADRB1MYLK4
SCHEMBL8515459 0.82 PRKD1 (0.46) DKK1ROCK2ADRB1MYLK4STK17A
Hydrochloric Acid SCHEMBL8512525 0.82 ROCK2 (0.41) KMODKK1ROCK2ADRB1MYLK4
Hydrochloric Acid SCHEMBL8511580 0.82 ROCK2 (0.41) KMODKK1ROCK2ADRB1MYLK4
SCHEMBL8512406 0.79 KMO (0.58) KMOPDE4D
SCHEMBL8515830 0.77 PRKD1 (0.45) DKK1ROCK2ADRB1MYLK4STK17A
SCHEMBL8512423 0.76 ADRB1 (0.42) DKK1ROCK2ADRB1MYLK4STK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO claimed
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed