SCHEMBL8512423

SCHEMBL8512423

C=C(C)c1ccc(-c2ccnc(N3CCNCC3)n2)cc1C(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.42
ROCK2 O75116 6/20 0.40
PIK3CA P42336 1/20 0.39
DKK1 O94907 3/20 0.39
MYLK4 Q86YV6 3/20 0.38
STK17A Q9UEE5 3/20 0.38
CLK4 Q9HAZ1 1/20 0.37
TBK1 Q9UHD2 1/20 0.37
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
UBE2N P61088 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8511182 0.99 ADRB1 (0.41) ADRB1ROCK2PIK3CADKK1MYLK4
SCHEMBL8511972 0.84 DKK1 (0.39) ROCK2PIK3CADKK1CLK4
Hydrochloric Acid SCHEMBL8514429 0.83 DKK1 (0.38) ROCK2PIK3CADKK1CLK4
SCHEMBL8515183 0.81 ACHE (0.48) PIK3CATBK1
SCHEMBL8515830 0.78 PRKD1 (0.45) ADRB1ROCK2PIK3CADKK1MYLK4
SCHEMBL8511790 0.78 ROCK2 (0.41) ADRB1ROCK2PIK3CADKK1MYLK4
Hydrochloric Acid SCHEMBL8512525 0.77 ROCK2 (0.41) ADRB1ROCK2DKK1MYLK4STK17A
Hydrochloric Acid SCHEMBL8511580 0.77 ROCK2 (0.41) ADRB1ROCK2DKK1MYLK4STK17A
SCHEMBL8511121 0.76 KMO (0.46) ADRB1ROCK2DKK1MYLK4STK17A
SCHEMBL8515459 0.76 PRKD1 (0.46) ADRB1ROCK2DKK1MYLK4STK17A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012069852-A1 PHARMACEUTICAL COMPOUNDS AS INHIBITORS OF SPHINGOSINE KINASE ALMAC DISCOVERY LIMITED (GB) 2012-05-31 WO disclosed